Publications of Don M. Coltart

Papers Submitted

  1. Lim, D.; Coltart, D. M., "A Simple and Efficient Method for Asymmetric α-Alkylation and α,α-Bisalkylation", J. Am. Chem. Soc., 2007.

Journal Articles

  1. Lim, D.; Zhou, G.; Livanos, A. E.; Fang, F.; Coltart, D. M., "MgBr2⋅OEt2-Promoted Coupling of Ketones and Activated Acyl Donors via Soft Enolization: A Practical Synthesis of 1,3-Diketones", Synthesis, (in press).
  2. Zhou, G.; Yost, J. M.; Sauer, S.; Coltart, D. M., "A Facile and Efficient Anti-Selective Four-Component Direct Aldol Addition via Chemoselective Thioester Enolate Formation", Org. Lett., 2007, 9, 4663-4665.
  3. Zhou, G.; Yost, J. M.; Coltart, D. M., "A Direct Aldol Addition of Simple Thioesters Employing Soft Enolization.", Synthesis, 2007, 478-482 (Invited paper.).
  4. Lim, D.; Fang, F.; Zhou, G.; Coltart, D. M, "Direct Carbon–Carbon Bond Formation via Soft Enolization: A Facile and Efficient Synthesis of 1,3-Diketones", Org. Lett., 2007, 9, 4139-4142.
  5. Yost, J.M., Zhou, G., and Coltart, D.M., "A Facile and Efficient Direct Aldol Addition of Simple Thioesters", Org. Lett., 2006, 8, 1503-1506 (Featured in Synfacts, September 2006, 591.).
  6. Clive, Derrick L. J.; Hisaindee, Soleiman; Coltart, Don M., "Derivatized Amino Acids Relevant to Native Peptide Synthesis by Chemical Ligation and Acyl Transfer", Journal of Organic Chemistry, 2003, 68(24), 9247-9254.
  7. Coltart, Don ; Danishefsky, Samuel J., "Novel Synthetic Approach to the 8,10-Dimethyl anti-syn-anti-Perhydrophenanthrene Skeleton", Organic Lett., 2003, 5(8), 1289-1292.
  8. Keding, S.J., Endo, A., Biswas, K., Zatorski, A., Coltart, D.M., Danishefsky, S.J., "Hydroxynorleucine as a Glycosyl Acceptor is an Efficient Means for Introducting Amino Acid Functionality into Complex Carbohydrates", Tetrahedron Lett., 2003, 44, 3413-3416.
  9. Ragupathi, Govindaswami; Coltart, Don M.; Williams, Lawrence J.; Koide, Fusataka; Kagan, Ella; Allen, Jennifer; Harris, Christina; Glunz, Peter W.; Livingston, Philip O.; Danishefsky, Samuel J., "On the power of chemical synthesis: immunological evaluation of models for multiantigenic carbohydrate-based cancer vaccines.", Proceedings of the National Academy of Sciences (USA), 2002, 99(21), 13699-13704.
  10. Coltart, Don M.; Royyuru, Ajay K.; Williams, Lawrence J.; Glunz, Peter W.; Sames, Dalibor; Kuduk, Scott D.; Schwarz, Jacob B.; Chen, Xiao-Tao; Danishefsky, Samuel J.; Live, David H., "Principles of Mucin Architecture: Structural Studies on Synthetic Glycopeptides Bearing Clustered Mono-, Di-, Tri-, and Hexasaccharide Glycodomains", J. Am Chem Soc., 2002, 124(33), 9833-9844.
  11. Clive, D.L., Coltart, D.M., Zhou, Y., de Lima, D.P., Yang, H., Lewanczuk, R.Z., "Synthesis of the Naturally Occuring ACE Inhibitors (-)-A58365A and (-)-A58365B, and of an Unnatural but Biologically Active Analog", 28th series, Actualité de Chimie Thérapeutique, French Society of Medicinal Chemistry, 2002, 21-50.
  12. Ragupathi, G., Deshpande, P.P., Coltart, D.M., Kim, H.J., Williams, L.J., Danishefsky, S.J., Livingston, P.O., "Constructing an Adenocarcinoma Vaccine: Immunization of Mice with Synthetic KH-1 Nonasaccharide Stimulates Anti-KH-1 and Anti-Ley Antibodies", Intl. J. Cancer, 2002, 99, 207-212.
  13. Biswas, K., Coltart, D.M., Danishefsky, S.J.,, "Construction of Carbohydrate-Based Antitumor Vaccines: Synthesis of Glycosyl Amino Acids by Olefin Cross-Metathesis", Tetrahedron Lett., 2002, 43, 6107-6110.
  14. D.M. Coltart, "Peptide segment coupling by prior ligation and proximity-induced intramolecular acyl transfer", Tetrahedron, 2000, 56(22), 3449-3491.
  15. Clive, D.L., Coltart, D.M., Zhou, Y, "Synthesis of the Angiotensin-Converting Enzyme Inhibitors (-)-A58365A and (-)-A58365B from a Common Intermediate", J. Org. Chem., 1999, 64, 1447-1454.
  16. Pelisson, M.M., da Silva, G.V.J., Clive, D.L.J., Coltart, D.M., Hof, F.A., "Studies on the Preparation of a,4-Disubstituted 2-Methoxypyridines", J. of Heterocycl. Chem, 1999, 36, 653-658.
  17. Clive, D.L.,J. and Coltart, D.M., "Synthesis of the Angiotensin-Converting Enzyme Inhibitor (±)-A58365A", Tetrahedron Lett., 1998, 39, 2519-2522.
  18. Coltart, D.M. and Charlton, J.L., "The Aymmetric Synthesis of Aryltetralin Lignans: (-)-Isolariciresinol Dimethyl Ether and (-)-Deoxysikkimotoxin", Can. J. Chem, 1996, 74, 88-94.